Source: San Jose Mercury News Contact: Pubdate: Wed, 22 Oct 1997 NOTE: From our newshawk: At the recent Drug Policy Foundation conference, Dr. John Morgan, a toxicologist, remarked on the irony of the St. John's wort craze. We know very little about the safety of this herb that is widely available at health food stores. Yet cannabis, which is a safely consumed herb about which we know a great deal, is illegal and people are being imprisoned for using it. Herb being used for depression BY SUSAN OKIE Washington Post CONSUMERS are snapping up St. John's wort preparations from the shelves of supermarkets and healthfood stores. During the month of July, after ``20/20'' aired a segment about psychiatrist Harold H. Bloomfield's book, ``Hypericum and Depression,'' Americans spent $2.5 million on extracts of the herb, according to Bob Bidlingmeyer, vice president of Lichtwer Pharma USA. Doctors uneasy Many doctors are uneasy that so many people are using St. John's wort to treat themselves, particularly if they are combining it with other medications. Una McCann, chief of the anxiety disorders unit at the National Institute of Mental Health, said she now routinely asks patients in her clinic if they are taking supplements or herbal products. ``I never would have asked that before,'' she said. Predicting which drugs might interact dangerously with St. John's wort is complicated because scientists still don't know exactly how the herb works. Walter Mueller, director of the Institute of Pharmacology at the University of Frankfurt in Germany, said his research in rats and mice shows that hypericum extract acts similarly to the antidepressants Zoloft and Prozac, blocking the ``reuptake'' by cells of a chemical called serotonin that carries messages between nerves in the brain. Thus, when serotonin is released at nerve endings, it hangs around longer and over several weeks, this in turn produces changes in the number of serotonin receptors, molecules on nerve surfaces that respond to the chemical message. He said this gradual change in receptors may be part of the reason why it often takes several weeks for hypericum as well as some other antidepressants to take effect. How it works But in addition to blocking serotonin reuptake, Mueller said, hypericum extract also blocks reuptake of the chemical messengers dopamine and norepinephrine. This nearly equal effect on three distinct messenger systems in the brain ``has never been shown for any of the other antidepressants,'' he said. Some psychiatrists said an interaction between Zoloft and St. John's wort may cause dangerous rise in blood pressure. They said people taking antidepressants or other prescription drugs should not stop them suddenly and should not try St. John's wort without consulting a physician. For people with mild depressive symptoms who are not taking any prescription drugs, opinion is divided. Mueller cautions that the herbal extract does not work for everyone. Bloomfield's book suggests the dose used in Germany 300 milligrams of hypericum extract three times a day and contains information about specific products and possible side effects, including indigestion, allergic reactions, tiredness, restlessness and a theoretical risk (seen in animals but so far not in humans) of severe skin reactions after sun exposure. Published Wednesday, October 22, 1997, in the San Jose Mercury News