Source: Washington Post (DC) Copyright: 1998 The Washington Post Company Pubdate: Sun, 29 Nov 1998 Page: C01 Contact: http://washingtonpost.com/wp-srv/edit/letters/letterform.htm Website: http://www.washingtonpost.com/ Author: Wayne Hall Note: Wayne Hall is executive director of the National Drug and Alcohol Research Centre in Sydney, Australia. Related: http://www.mapinc.org/drugnews/v98.n1041.a04.html http://www.mapinc.org/drugnews/v98.n1041.a05.html http://www.mapinc.org/drugnews/v98.n1041.a06.html PAST THE SMOKE SCREEN Forget Your Presumptions. Medical Marijuana Needs the Same Scrutiny as Any Other Drug More closely associated with the likes of Cheech and Chong than with chemotherapy, with pot parties than with pain relief, marijuana is mostly thought of as an illegal substance. The claim that it might be useful in treating a variety of medical conditions typically provokes two divergent and equally unrealistic responses: Opponents argue that the plant offers little or no therapeutic benefit; advocates see it as a powerfully effective drug that no one should be denied. In the United States, the debate about the medical use of marijuana has become mired in the political arena. Voters in five states (Alaska, Arizona, Nevada, Oregon and Washington) recently approved medical marijuana initiatives--despite arguments from federal officials, police chiefs and some state legislatures that, at best, such a move promotes a mixed message and, at worst, represents a thinly veiled attempt to legalize marijuana for recreational use. (In the District, a congressional amendment has blocked election officials from even counting the votes on Initiative 59, a medical marijuana referendum that was on the November ballot; the standoff is now in the hands of a federal judge.) Lost in the political haze--and in the popular fantasies about the drug's potency--are the complexities in evaluating marijuana's usefulness as medicine. The same has been true, in my experience, in trying to assess the health risks of recreational marijuana use, an issue I addressed in an article earlier this month in the Lancet, the British medical journal. Putting politics aside for the moment, let's suppose that prescribing marijuana in its plant form became legal. How likely would doctors be to use it? Where does it belong in the array of medications now available for treating pain or the nausea that often accompanies chemotherapy? In short, would it benefit or hurt patients? Physicians and researchers aren't nearly as certain about the answers to these critical questions as are the advocates and opponents. Definitive answers are hard to come by, partly because of the absence of scientific research on the drug's efficacy. Since much of the world's research on drugs takes place in the United States, the Drug Enforcement Agency's classification of the marijuana plant (cannabis sativa) as having "no medical use" has made it difficult to do the clinical trials that usually provide the best information on a drug's benefits and side effects. The very nature of marijuana makes it hard to test in clinical trials. Unlike drugs such as morphine or Viagra, marijuana is a crude plant product that contains a complex and varied mixture of 60 substances known as cannabinoids. Before a drug can be registered, the FDA requires that it be a pure substance of known chemical structure that can be shown in controlled trials to be safe and effective at particular doses in the treatment of particular diseases. Physicians have long had the authority to prescribe painkillers, but clinical trials have helped clarify the risks and benefits of particular doses. So, for example, physicians know they can give patients suffering acute pain an injection of 2.5 to 15 milligrams of morphine, and that their pain will be relieved for several hours with a low risk of adverse effects. The point here isn't that marijuana is particularly dangerous. All drugs pose dangers--that is, all drugs contain risks that must be identified and weighed. And at this point, we don't know as much about the medical risks of marijuana as we should. The difficulties of evaluating the therapeutic uses of marijuana are amplified by the dizzying variety of medical conditions for which its more enthusiastic advocates claim it is useful. They include the nausea and vomiting caused by chemotherapy, AIDS-related wasting caused by loss of appetite, multiple sclerosis, paraplegia, some forms of chronic pain, glaucoma and asthma. For about a decade, doctors have been able to prescribe one of marijuana's constituents, the cannabinoid tetrahydrocannabinol or THC, which is the ingredient responsible for many of marijuana's psychological effects, such as relaxation and euphoria. But THC hasn't proven to be a particularly useful drug. Now marketed in pill form under the trade name Marinol, THC can be used to treat the nausea and vomiting experienced by chemotherapy patients and to stimulate appetite in AIDS patients. These are the only medical uses of cannabinoids that are supported thus far by evidence from controlled clinical trials. The DEA has argued that the registration of Marinol obviates the need to register marijuana itself for medical use. Despite having been available in the United States for more than a decade, Marinol is rarely used to treat nausea and vomiting because other drugs have become available that have proven to be effective, such as ondansetron and granisetron. And those patients who have taken Marinol as an appetite stimulant have found it difficult to get the dosage right; the effects of THC are delayed when taken orally, making it hard to regulate the amount needed to achieve the desired therapeutic benefit. Some patients report receiving too little THC to relieve their symptoms; others, in particular those who have no experience with marijuana, report feeling tired, lethargic and drowsy after taking the medication. These sorts of reactions to Marinol contrast sharply with the anecdotal evidence from AIDS patients who have smoked marijuana. Some of these patients have reported marked improvements. Smoking marijuana allowed them to use as much or as little of the drug as they felt they needed to relieve their symptoms. Experiences like these, reported by Harvard psychiatrist Lester Grinspoon and his legal colleague James B. Bakalar in their 1997 book "Marijuana, The Forbidden Medicine," led them to conclude that marijuana smoking should be allowed for medical reasons. Some advocates also say that smoking is a more sociable way of using medications and might have advantages over popping a pill--factors that don't normally figure into regulatory decisions about which drugs to approve for medical use. But in most developed countries, medical societies and government regulators have typically rejected medical marijuana smoking. Many doctors are uncomfortable with promoting any form of smoking, given the risks of smoking tobacco products. They also point out that the burning of marijuana and tobacco produces many of the same cancer-causing substances (although marijuana does not contain nicotine). The cancer risk of marijuana may be minor for the occasional user, but it becomes a more important question if marijuana is used to treat a chronic health problem such as glaucoma or multiple sclerosis--when a patient might smoke it several times a day for months or years. In the case of AIDS patients, smoking marijuana may stimulate appetite but it may also further depress their immune systems, leaving them more vulnerable to opportunistic infections. The plant also may be contaminated with microorganisms that can be life-threatening for patients whose immune systems are already compromised. For many doctors, the central question is: Should we insist that patients use only a pure drug, the effects of which are difficult to control, or should we allow the medical use of smoked marijuana with all its drawbacks? Neither alternative is ideal. But then, no drug is perfect; all have side effects, and the side effects of marijuana are arguably no worse than those of other therapeutic drugs. If marijuana were not an illegal drug, widely used for recreational reasons, the choice would be left primarily to doctors and their patients. Expert opinion may be changing a little on this issue. A panel of experts convened by the National Institutes of Health to look into these sorts of questions reported last year that smoking marijuana may be useful for treating a number of conditions--although it may not be better than other medications. In Britain, a subcommittee of the House of Lords suggested in a report released earlier this month that the medical value of smoked marijuana should be explored. It recommended that if smoked marijuana proved to be therapeutically better than oral THC, then methods should be developed to inhale cannabinoids without the potentially harmful byproducts that are produced when the leaf is burned. Ironically enough, the tobacco industry's recent attempts to develop a "smokeless" nicotine delivery system might provide the means. Other obstacles would arise if marijuana smoking were approved for medical purposes. Pharmaceutical companies do not have any commercial incentive to register and market a non-patentable, naturally occurring plant product. Similar disincentives delayed, for several years, the use of naturally occurring pure Lithium salts for the treatment of manic-depressive illness. The key to moving the current debate forward rests in a better scientific understanding of the way in which marijuana and its constituent cannabinoids act in the human brain. In the early 1990s, researchers identified a receptor in animal and human brains that responds specifically to THC, as well as a naturally occurring analog of THC, anandamide. These discoveries have led to the synthesis of new substances that are chemically related to THC and other cannabinoids. Some of these--and others yet to be synthesized--may produce the desired therapeutic effects without the side effects pursued by recreational users. Not all the consequences of research on the chemistry and pharmacology of cannabinoids may be desirable. If, for example, it proved easy to synthesize cannabinoids that had psychoactive effects like THC, then the opportunities for recreational cannabinoid use would probably increase markedly. Similarly, if water-soluble cannabinoids are developed for more efficient oral use, they could also be injected, substantially increasing the potential for abuse of cannabinoids in much the same way that cocaine or heroin have done for the coca plant or opium poppy. The price we pay for medically useful cannabinoid drugs may be more dangerous synthetic derivatives of marijuana. The issue of whether to fund clinical trials remains highly controversial; even if trials were to be funded, the regulatory process would take five to 10 years, at best. Advances in our understanding of cannabinoid chemistry could dramatically change what we think about marijuana's usefulness. Meanwhile, I would hazard three predictions about the medical use of marijuana and cannabinoid drugs over the next 20 years: First, if marijuana has a medical role, it will be more akin to an herbal remedy than mainstream treatment. Second, drugs derived from cannabis will have a medical role but a much more modest one than their more enthusiastic advocates would have us believe. And third, the development of new and better drugs may make the current battle over medical marijuana seem like a puzzling--but fascinating--historical curiosity. - --- Checked-by: Richard Lake